WQQ-345
WQQ-345 is a BCAT1 inhibitor (IC50: 10.8 mM) that suppresses glycolysis by reducing α-KG and downregulating PFKP and LDHA, while increasing H3K27me3 in vitro. It has also demonstrated antitumor efficacy in a 67R cell xenograft mouse model, supporting its use in cancer metabolism research.
Product Specifications
Field of Research
Epigenetics & Chromatin, Metabolism Research
Molecular Formula
C10H17NO2
Molecular Weight
183.25
Storage Conditions
-20°C
Notes
For research use only.
Available Sizes
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