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WQQ-345

WQQ-345 is a BCAT1 inhibitor (IC50: 10.8 mM) that suppresses glycolysis by reducing α-KG and downregulating PFKP and LDHA, while increasing H3K27me3 in vitro. It has also demonstrated antitumor efficacy in a 67R cell xenograft mouse model, supporting its use in cancer metabolism research.

Product Specifications

Field of Research

Epigenetics & Chromatin, Metabolism Research

Molecular Formula

C10H17NO2

Molecular Weight

183.25

Storage Conditions

-20°C

Notes

For research use only.

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