MNI137
MNI137 is a potent and selective negative allosteric modulator for group II mGluRs. MNI137 has IC50s values of 8.3 and 12.6 nM for human and rat mGlu2 inhibition of glutamate-induced calcium mobilization.
Product Specifications
CAS Number
946619-21-2
Purity
>98%
Smiles
N#CC1N=CC=C (C2CCC (=O) NC3=CC (=CC=C3N=2) Br) C=1
Molecular Formula
C16H11BRN4O
Molecular Weight
355.188741922379
Notes
For research use only.
Available Sizes
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