VU6008677
VU6008677 is a potent and selective positive allosteric modulator (PAM) of the human M4 muscarinic receptor (EC50 = 120 nM) . This research compound is utilized in vitro and in vivo to investigate the therapeutic potential of M4 modulation for central nervous system disorders, though it exhibits high metabolic clearance and plasma protein binding.
Product Specifications
CAS Number
2170550-99-7
Field of Research
Metabolism Research, Neuroscience
Smiles
ClC1=C (N=C2OC=3C (=NC=NC3C2=C1C) NC4CC4) C
Molecular Formula
C14H13ClN4O
Molecular Weight
288.73
Storage Conditions
-20°C
Notes
For research use only.
Available Sizes
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