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HA2AAR antagonist 1

Compound 4a (hA2AAR antagonist 1) is a potent and selective human A2A adenosine receptor antagonist with a Ki of 5 nM. It is a valuable research tool in immuno-oncology, used in both in vitro and in vivo studies to investigate adenosine-mediated immunosuppression in the tumor microenvironment.

Product Specifications

CAS Number

2842150-81-4

Field of Research

Neuroscience, Pharmacology & Drug Discovery

Smiles

C (#CCCCC) C1=NC2=NC (=NC (N) =C2N1) C=3OC=CC3

Molecular Formula

C15H15N5O

Molecular Weight

281.31

Storage Conditions

-20°C

Notes

For research use only.

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