ER degrader 9
Compound 1 (ER degrader 9) is a potent bifunctional degrader of the estrogen receptor, demonstrating a DC50 of ≤10 nM in MCF-7 breast cancer cells. It is a valuable research tool for investigating ERα biology and targeted protein degradation in breast cancer models, both in vitro and in vivo.
Product Specifications
CAS Number
3023359-75-0
Field of Research
Metabolism Research, Pharmacology & Drug Discovery
Smiles
OC=1C=C2C ([C@H] ([C@H] (CC2) C3=CC=CC=C3) C4=CC=C (C=C4) N5CCC (CN6CCN (C (/C (=C\C (C) (C) C) /C#N) =O) CC6) CC5) =CC1
Molecular Formula
C40H48N4O2
Molecular Weight
616.83
Storage Conditions
-20°C
Notes
For research use only.
Available Sizes
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