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PDHK-IN-7

PDHK-IN-7 (compound 32) is a potent pyruvate dehydrogenase kinase (PDK) inhibitor with an IC50 of 17 nM. It activates pyruvate dehydrogenase (PDH) in vitro and has demonstrated in vivo efficacy by reducing blood glucose levels in Zucker obese rat models, supporting research in metabolic disorders like diabetes and obesity.

Product Specifications

CAS Number

1220965-73-0

Field of Research

Metabolism Research

Smiles

FC (F) (F) C1 (O) C=2C=CC=CC2C3=C (C=C (C=C31) C) C=4C=NN (C4) CCO

Molecular Formula

C20H17F3N2O2

Molecular Weight

374.36

Storage Conditions

-20°C

Notes

For research use only.

Available Sizes

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