PDHK-IN-7
PDHK-IN-7 (compound 32) is a potent pyruvate dehydrogenase kinase (PDK) inhibitor with an IC50 of 17 nM. It activates pyruvate dehydrogenase (PDH) in vitro and has demonstrated in vivo efficacy by reducing blood glucose levels in Zucker obese rat models, supporting research in metabolic disorders like diabetes and obesity.
Product Specifications
CAS Number
1220965-73-0
Field of Research
Metabolism Research
Smiles
FC (F) (F) C1 (O) C=2C=CC=CC2C3=C (C=C (C=C31) C) C=4C=NN (C4) CCO
Molecular Formula
C20H17F3N2O2
Molecular Weight
374.36
Storage Conditions
-20°C
Notes
For research use only.
Available Sizes
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