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LGB321

LGB321 is a potent and selective PIM2 kinase inhibitor that suppresses the proliferation of PIM2-dependent multiple myeloma cells. It effectively inhibits key oncogenic pathways, including mTORC1 signaling and BAD phosphorylation, making it a valuable tool for in vitro and in vivo studies of hematological malignancies.

Product Specifications

CAS Number

1210417-75-6

Field of Research

Signal Transduction

Smiles

N (C (=O) C=1N=C (C (F) =CC1) C2=C (F) C=CC=C2F) C=3C (=CC=NC3) N4C[C@H] (C) [C@@H] (O) [C@H] (N) C4

Molecular Formula

C23H22F3N5O2

Molecular Weight

457.45

Storage Conditions

-20°C

Notes

For research use only.

Available Sizes

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