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DA-023

DA-023 (Compound 4) is a potent and selective positive allosteric modulator (PAM) for the EAAT2 transporter, with an EC50 of 1 nM. This small molecule is a valuable research tool for investigating glutamate clearance in models of neurological disorders, both in cellular assays and animal studies.

Product Specifications

CAS Number

2585643-97-4

Field of Research

Metabolism Research

Smiles

C (C=1N (CCC2=CC=CC=C2) N=NN1) (N3CCN (C) CC3) C=4C=CC=NC4

Molecular Formula

C20H25N7

Molecular Weight

363.46

Storage Conditions

-20°C

Notes

For research use only.

Available Sizes

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