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INY-05-040

INY-05-040 is a potent, pan-AKT degrader that rapidly depletes all AKT isoforms, blocking downstream signaling and suppressing proliferation across a broad panel of cancer cell lines. Its utility extends to in vitro mechanistic studies and in vivo preclinical research targeting PI3K/AKT-driven cancers.

Product Specifications

CAS Number

2503018-29-7

Field of Research

Pharmacology & Drug Discovery, Signal Transduction

Smiles

C[C@H]1C2=C (N=CN=C2[C@H] (O) C1) N3CCN (C ([C@H] (CNCCCCCCCCCCC (N[C@H] (C (=O) N4[C@H] (C (N[C@@H] (C) C5=CC=C (C=C5) C=6SC=NC6C) =O) C[C@@H] (O) C4) C (C) (C) C) =O) C7=CC=C (Cl) C=C7) =O) CC3

Molecular Formula

C55H76ClN9O6S

Molecular Weight

1026.77

Storage Conditions

-20°C

Notes

For research use only.

Available Sizes

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