LASSBio-873
LASSBio-873 is an orally bioavailable, brain-penetrant small molecule agonist of muscarinic acetylcholine receptors (mAChRs) . It demonstrates significant analgesic efficacy in models of acute and inflammatory pain, an effect mediated through M2 receptor activation as shown by antagonist studies. This profile makes it a valuable research tool for investigating cholinergic pathways in pain modulation.
Product Specifications
CAS Number
873694-54-3
Field of Research
Neuroscience, Pharmacology & Drug Discovery
Purity
98.83% (May vary between batches)
Smiles
O=C1C2=CN=C3C (C (C) =NN3C4=CC=CC=C4) =C2C (N1C5=CC=C ([N+] ([O-]) =O) C=C5) =O
Molecular Formula
C21H13N5O4
Molecular Weight
399.36
Storage Conditions
-20°C
Notes
For research use only.
Available Sizes
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