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MAT2A-IN-13

MAT2A-IN-13 is an orally bioavailable, potent inhibitor of methionine adenosyltransferase 2A (MAT2A) . It shows promising in vivo efficacy in MTAP-deleted xenograft models, supporting its use as a research tool for investigating synthetic lethality in MTAP-deficient cancers.

Product Specifications

CAS Number

2851449-24-4

Field of Research

Epigenetics & Chromatin, Signal Transduction

Smiles

O=C1C (=C2N (C (NC3CC3) =N1) C=CC (C (F) (F) F) =C2) C4=C (F) N=CC=C4

Molecular Formula

C17H12F4N4O

Molecular Weight

364.3

Storage Conditions

-20°C

Notes

For research use only.

Available Sizes

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