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ERAP1 modulator-1

ERAP1 modulator-1 (Compound 1) is a potent small molecule inhibitor of endoplasmic reticulum aminopeptidase 1, exhibiting an IC50 below 250 nM. This compound is a valuable research tool for studying ERAP1's role in antigen processing, peptide trimming, and its implications in autoimmune diseases and cancer immunotherapy in both cellular and biochemical assays.

Product Specifications

CAS Number

2766036-51-3

Field of Research

Cell Biology, Metabolism Research

Molecular Formula

C23H23F3N2O5S

Molecular Weight

496.5

Storage Conditions

-20°C

Notes

For research use only.

Available Sizes

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