EZH2-IN-22
EZH2-IN-22 is a highly potent small molecule inhibitor of EZH2, demonstrating sub-nanomolar IC50 values against both wild-type and mutant (Y641N, Y641F) forms. Its robust antiproliferative activity supports its use in vitro for epigenetic cancer research and in vivo for studying oncogenic mechanisms in preclinical models.
Product Specifications
CAS Number
2766231-05-2
Field of Research
Epigenetics & Chromatin
Smiles
C (=C\C (O) =O) \C (O) =O.N (CC) (C1=C (C) C (C (NCC2=C (C) C=C (C) NC2=O) =O) =CC (O[C@@H]3C[C@H] (C3) N4CCCCC4) =C1) C5CCOCC5
Molecular Formula
C36H50N4O8
Molecular Weight
666.8
Storage Conditions
-20°C
Notes
For research use only.
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