Anticancer agent 258
Anticanceragent 258 is a potent imidazotriazole-based modulator of Nurr1 (EC50=63 nM in N2A cells) and Nur77 (IC50=0.1 pM in HEK293 cells) . This small molecule is a valuable research tool for investigating nuclear receptor function in cancer biology, metabolic disease, and neurological disorder models, both in vitro and in vivo.
Product Specifications
CAS Number
2891984-12-4
Field of Research
Pharmacology & Drug Discovery
Smiles
FC=1C=CC (=CC1) C=2N=C3N (N2) C=C (C=4C=CC=C (F) C4) N3C
Molecular Formula
C17H12F2N4
Molecular Weight
310.3
Storage Conditions
-20°C
Notes
For research use only.
Available Sizes
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