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PDE4B/D-IN-3

PDE4B/D-IN-3 (example 22) is a potent and selective PDE4 inhibitor, demonstrating IC50 values of 0.071 nM for PDE4B2 and 0.09 nM for PDE4D. This compound is a valuable research tool for studying PDE4 biology in cellular assays and animal models of inflammation and central nervous system disorders.

Product Specifications

CAS Number

3034683-69-4

Field of Research

Metabolism Research, Signal Transduction

Smiles

N (C1=C2C (=NC (=N1) N3CC=4C (CC3) =CC (=CC4) C=5N=CC=CN5) CCS2=O) C6CCOCC6

Molecular Formula

C24H26N6O2S

Molecular Weight

462.57

Storage Conditions

-20°C

Notes

For research use only.

Available Sizes

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