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HPK1-IN-2 dihydrochloride

HPK1-IN-2 dihydrochloride is a potent, orally bioavailable small molecule inhibitor of HPK1 (IC50 <0.05 μM) with additional activity against Lck and Flt3 kinases. This compound has demonstrated significant antitumor efficacy in research models, supporting its investigation in oncology and immunology for both in vitro and in vivo studies.

Product Specifications

CAS Number

2375595-72-3

Field of Research

Cardiovascular Research, Signal Transduction

Smiles

NC1=C (C=2NC=3C (N2) =CC=C (C3) N4CCN (C) CC4) C (=O) NC5=C1C=CS5.Cl

Molecular Formula

C19H22Cl2N6OS

Molecular Weight

453.39

Storage Conditions

-20°C

Notes

For research use only.

Available Sizes

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