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(R) -IDO/TDO-IN-1

(R) -IDO/TDO-IN-1 is a potent dual inhibitor of indoleamine-2,3-dioxygenase (IDO) with favorable pharmacokinetics. It shows single-agent anti-tumor activity in the MC38 mouse xenograft model and demonstrates synergistic efficacy in combination with anti-PD-1 therapy, supporting its use in immuno-oncology research.

Product Specifications

CAS Number

2033173-00-9

Field of Research

Metabolism Research

Smiles

FC1=C2[C@H] (N3C (C2=CC=C1) =CN=C3) C4CCN (CC4) C5=CC=C (C=C5) C6=CN (C) N=C6

Molecular Formula

C25H24FN5

Molecular Weight

413.49

Storage Conditions

-20°C

Notes

For research use only.

Available Sizes

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