RS-127445 maleate
RS-127445 maleate is a potent and selective 5-HT2B receptor antagonist with a pKi of 9.5 and demonstrated oral bioavailability. It is a valuable research tool for investigating serotonin receptor function in both in vitro binding assays and in vivo models of cardiovascular and fibrotic diseases.
Product Specifications
CAS Number
199864-88-5
Smiles
C (=C\C (O) =O) \C (O) =O.FC=1C2=C (C (=CC1) C=3C=C (C (C) C) N=C (N) N3) C=CC=C2
Molecular Formula
C21H20FN3O4
Molecular Weight
397.406
Storage Conditions
-20°C
Notes
For research use only.
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