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Mps1-IN-10

Mps1-IN-6 (Compound 9) is a potent and selective Mps1 kinase inhibitor with an IC50 of 6.4 nM. It demonstrates robust anti-proliferative activity against breast cancer cells in vitro and has shown promising anti-tumor efficacy in relevant in vivo models, supporting its use in oncology research.

Product Specifications

CAS Number

2489220-49-5

Field of Research

Signal Transduction

Smiles

N (C1=C2C (=NC (NC3=C (OC) C=C (C=C3) N4C (=O) CCC4) =N1) NC=C2C#N) C5CCCCC5

Molecular Formula

C24H27N7O2

Molecular Weight

445.52

Storage Conditions

-20°C

Notes

For research use only.

Available Sizes

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