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PF15 TFA

PF15 TFA is a CRBN-based PROTAC that selectively degrades FLT3-ITD with a DC50 of 76.7 nM. It inhibits proliferation and downstream signaling in FLT3-ITD+ cells and has demonstrated efficacy in reducing tumor growth in murine models of acute myeloid leukemia.

Product Specifications

Field of Research

Cardiovascular Research, Immunology & Inflammation, Pharmacology & Drug Discovery, Signal Transduction

Molecular Formula

C46H50F3N13O8

Molecular Weight

969.97

Storage Conditions

-20°C

Notes

For research use only.

Available Sizes

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