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SJ1008030 TFA

SJ1008030 (compound 8) TFA is a potent and selective PROTAC degrader of JAK2. It demonstrates anti-leukemic activity in vitro, inhibiting the proliferation of MHH-CALL-4 cells with an IC50 of 5.4 nM, supporting its utility in hematological cancer research.

Product Specifications

Field of Research

Cardiovascular Research, Epigenetics & Chromatin, Immunology & Inflammation, Pharmacology & Drug Discovery, Signal Transduction, Stem Cell & Developmental Biology

Molecular Formula

C44H44F3N13O9S

Molecular Weight

987.96

Storage Conditions

-20°C

Notes

For research use only.

Available Sizes

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