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PRMT5-IN-25

PRMT5-IN-25 is a highly potent and selective PRMT5 inhibitor with a Ki of 0.06 nM. This compound demonstrates robust antiproliferative activity in cellular assays and is a valuable chemical probe for investigating PRMT5 function in oncology and epigenetics research, both in vitro and in vivo.

Product Specifications

CAS Number

2691869-82-4

Field of Research

Epigenetics & Chromatin

Smiles

C (N (CC1=CC=C (C (F) (F) F) C=N1) [C@H] (C) C=2N=CC=CN2) (=O) C3=CC4=C (C=C3) N=C (N) C (C) =C4

Molecular Formula

C24H21F3N6O

Molecular Weight

466.46

Storage Conditions

-20°C

Notes

For research use only.

Available Sizes

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