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STX-478

STX-478 is a brain-penetrant, selective PI3Kα inhibitor for research use. It demonstrates anticancer activity in preclinical models, inhibiting tumor growth in studies relevant to breast cancer and other solid tumors.

Product Specifications

CAS Number

2883540-92-7

Product Name Alternative

PI3Kα

Field of Research

Signal Transduction

Purity

98.31% (May vary between batches)

Solubility

DMSO:100 mg/mL (249.2 mM) ;10% DMSO+40% PEG300+5% Tween 80+45% Saline:5 mg/mL (12.46 mM)

Smiles

[C@H] (NC (NC=1C=NC (N) =NC1) =O) (C (F) (F) F) C2=C (C) C=3C (O2) =C (F) C=C (F) C3

Molecular Formula

C16H12F5N5O2

Molecular Weight

401.29

Storage Conditions

-20°C

Notes

For research use only.

Available Sizes

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