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MHJ-627

MHJ-627 is a potent and selective ERK5 (MAPK7) inhibitor with an IC50 of 0.91 μM. It upregulates tumor suppressor and anti-metastatic gene expression, inducing cancer cell death in vitro. This small molecule is a valuable chemical probe for studying ERK5 signaling in oncology research, including investigations into metastasis and apoptosis.

Product Specifications

Field of Research

Signal Transduction

Molecular Formula

C34H45BrN2O3

Molecular Weight

609.64

Storage Conditions

-20°C

Notes

For research use only.

Available Sizes

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