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WCA-814

WCA-814 is a bifunctional small molecule that acts as an androgen receptor antagonist and Hsp90 inhibitor conjugate. It effectively degrades both full-length AR and the splice variant AR-V7, demonstrating potent in vitro cytotoxicity in prostate cancer cell lines such as LNCaP and 22Rv1.

Product Specifications

Field of Research

Metabolism Research

Molecular Formula

C46H53ClN10O5

Molecular Weight

861.43

Storage Conditions

-20°C

Notes

For research use only.

Available Sizes

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