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CaSR antagonist-1

CaSR Antagonist-1 is a potent and selective calcium-sensing receptor (CaSR) inhibitor with an IC50 of 50 nM. It is a valuable research tool for studying CaSR function in vitro and in vivo, particularly in models of bone and mineral metabolism disorders such as osteoporosis.

Product Specifications

CAS Number

1219811-83-2

Field of Research

Pharmacology & Drug Discovery

Smiles

C (CC1=CC=CC=C1) N2C (=NC (C) =C (C2=O) C3=CC (=C (C) S3) C4=CC=CC=N4) C5=C (O) C (F) =CC=C5

Molecular Formula

C29H24FN3O2S

Molecular Weight

497.58

Storage Conditions

-20°C

Notes

For research use only.

Available Sizes

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