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PF-06478939

PF-06478939 is a potent peripheral agonist targeting oxytocin and vasopressin receptors with EC50 values of 0.01 nM and 0.078 nM, respectively. Its inability to cross the blood-brain barrier makes it a valuable tool for investigating the peripheral physiological roles of these receptors in cardiovascular, renal, and reproductive research using in vivo models.

Product Specifications

Field of Research

Metabolism Research, Pharmacology & Drug Discovery

Molecular Formula

C78H134N14O22S2

Molecular Weight

1684.11

Storage Conditions

-20°C

Notes

For research use only.

Available Sizes

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