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BMPR2-IN-1

BMPR2-IN-1 (Compound 8a) is a potent and selective BMPR2 inhibitor with a Kd of 83.5 nM. This small molecule is a valuable research tool for investigating the role of BMPR2 signaling in diseases such as pulmonary arterial hypertension, Alzheimer's disease, and cancer, in both cellular and animal models.

Product Specifications

Field of Research

Signal Transduction, Stem Cell & Developmental Biology

Smiles

O=C1C2=CC (NC3=CC=NC (NC4=CC=C (CCN1) C=C4) =N3) =NN2

Molecular Formula

C16H15N7O

Molecular Weight

321.34

Storage Conditions

-20°C

Notes

For research use only.

Available Sizes

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