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PROTAC TG2 degrader-2

PROTAC TG2 degrader-2 is a selective, competitive small molecule degrader of Transglutaminase 2 (TG2) with a Kd >100 μM. It has been shown to reduce TG2 protein levels and inhibit cell migration in ovarian cancer cell models, serving as a useful chemical probe for cancer biology and migration studies.

Product Specifications

Field of Research

Pharmacology & Drug Discovery, Protein Biochemistry

Molecular Formula

C47H57N9O6S

Molecular Weight

876.08

Storage Conditions

-20°C

Notes

For research use only.

Available Sizes

Frequently Asked Questions

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