HCYP3A4-IN-1

HCYP3A4-IN-1 (C6) is a potent, orally bioavailable competitive inhibitor of cytochrome P450 3A4, with an IC50 of 43.93 nM in HLMs. Its application is valuable for in vitro drug metabolism studies and in vivo pharmacokinetic interaction research, aiding the investigation of CYP3A4-mediated drug-drug interactions.