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DprE1-IN-6

DprE1-IN-6 (Compound 56) is a potent DprE1 inhibitor with anti-tuberculosis activity, showing a 1 μM MIC against Mtb H37Rv and efficacy against drug-resistant strains. It exhibits favorable pharmacokinetic properties, including high microsomal stability and medium clearance, supporting its utility in both in vitro and in vivo TB drug discovery research.

Product Specifications

Field of Research

Infectious Disease & Virology

Molecular Formula

C22H24N6O

Molecular Weight

388.47

Storage Conditions

-20°C

Notes

For research use only.

Available Sizes

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