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RORγ antagonist 1

RORγ antagonist 1 is a potent betulinic acid derivative functioning as a RORγ antagonist (K D = 0.18 μM) . It exhibits anti-proliferative activity in pancreatic cancer models, suppressing RAS/MAPK and AKT/mTORC1 pathways while inducing caspase-dependent apoptosis in vitro and in vivo.

Product Specifications

Field of Research

Metabolism Research, Pharmacology & Drug Discovery

Molecular Formula

C35H60N2O2

Molecular Weight

540.86

Storage Conditions

-20°C

Notes

For research use only.

Available Sizes

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