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MOR agonist-2

MOR agonist-2 (Compound 46) is a dual-activity small molecule functioning as a mu-opioid receptor (MOR) partial agonist (K i = 564 nM) and a dopamine D3 receptor (D3R) antagonist (K i = 7.26 nM) . This profile suggests potential for analgesia with a possibly reduced abuse liability, making it a candidate for research in neuropharmacology and pain management.

Product Specifications

Field of Research

Metabolism Research, Neuroscience, Pharmacology & Drug Discovery

Molecular Formula

C37H47Cl2N5O3

Molecular Weight

680.71

Storage Conditions

-20°C

Notes

For research use only.

Available Sizes

Frequently Asked Questions

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