MOR agonist-2
MOR agonist-2 (Compound 46) is a dual-activity small molecule functioning as a mu-opioid receptor (MOR) partial agonist (K i = 564 nM) and a dopamine D3 receptor (D3R) antagonist (K i = 7.26 nM) . This profile suggests potential for analgesia with a possibly reduced abuse liability, making it a candidate for research in neuropharmacology and pain management.
Product Specifications
Field of Research
Metabolism Research, Neuroscience, Pharmacology & Drug Discovery
Molecular Formula
C37H47Cl2N5O3
Molecular Weight
680.71
Storage Conditions
-20°C
Notes
For research use only.
Available Sizes
Frequently Asked Questions
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