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HCA/VEGFR-2-IN-3

HCA/VEGFR-2-IN-3 is a potent dual inhibitor targeting both carbonic anhydrase isoforms (hCA IX/XII) and VEGFR-2 kinase, with Ki values in the low nanomolar range. It demonstrates specific antiproliferative effects in VEGFR-2-overexpressing breast cancer cell lines, supporting its investigation in oncology research for tumor angiogenesis and acidosis.

Product Specifications

Field of Research

Cardiovascular Research, Cardiovascular Research; Cell Biology, Metabolism Research, Signal Transduction

Molecular Formula

C24H28N6O6S

Molecular Weight

528.58

Storage Conditions

-20°C

Notes

For research use only.

Available Sizes

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