BRD4 Inhibitor-10
Product Specifications
UNSPSC Description
BRD4 Inhibitor-10 is a potent BRD4-BD1 inhibitor extracted from patent WO2015022332A1, Compound II-25, has an IC50 of 8 nM[1].
Target Antigen
Epigenetic Reader Domain
Type
Reference compound
Related Pathways
Epigenetics
Field of Research
Cancer
Assay Protocol
https://www.medchemexpress.com/brd4-inhibitor-10.html
Purity
99.52
Solubility
DMSO : 125 mg/mL (ultrasonic)
Smiles
CN1C(C(C)=CC(C2=NC3=CN=C(C=C3N2[C@H](C4=CC=CC=C4)C)C5CCOCC5)=N1)=O
Molecular Weight
429.51
References & Citations
[1]Harald Engelhardt, et al. Pyridinones. WO2015022332A1.
Shipping Conditions
Room Temperature
Storage Conditions
-20°C, 3 years; 4°C, 2 years (Powder)
Product Datasheet
http://file.medchemexpress.com/batch_PDF/HY-117491/BRD4-Inhibitor-10-DataSheet-MedChemExpress.pdf
Product MSDS
http://file.medchemexpress.com/batch_PDF/HY-117491/BRD4-Inhibitor-10-SDS-MedChemExpress.pdf
Clinical Information
Phase 1
CAS Number
1660117-38-3
Available Sizes
Curated Selection
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