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NOX-6-18

NOX-6-18 (GPR132-B-160) is a potent and selective GPR132 antagonist. It exhibits insulinotropic effects and modulates macrophage activity in pancreatic islets, which has been studied in models of metabolic disease for its potential to reduce weight gain.

Product Specifications

CAS Number

898211-21-7

Product Name Alternative

GPR132, GPR132 antagonist 1, GPR132-B-160, NOX618

Field of Research

Metabolism Research, Pharmacology & Drug Discovery

Purity

99.29% (May vary between batches)

Solubility

DMSO:250 mg/mL (695.6 mM) ;10% DMSO+40% PEG300+5% Tween 80+45% Saline:3.3 mg/mL (9.18 mM)

Smiles

O=C (O) C=1OC=2C=CC (=CC2C1C) S (=O) (=O) NCCC=3C=CC=CC3

Molecular Formula

C18H17NO5S

Molecular Weight

359.4

Storage Conditions

-20°C

Notes

For research use only.

Available Sizes

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