RGH-122
RGH-122 (compound 43) is a potent, selective, and orally bioavailable hV1a receptor antagonist with sub-nanomolar affinity (K i 0.3 nM) . Its metabolic stability and pharmacological profile support its use in research exploring vasopressin V1a receptor function in cardiovascular, stress, and social behavior models, both in vitro and in vivo.
Product Specifications
CAS Number
2355304-05-9
Field of Research
Pharmacology & Drug Discovery
Smiles
ClC=1C=C2CC3 (CC=4N (C2=CC1) C (=NN4) [C@@H]5CC[C@@H] (OC6=CC=CC=N6) CC5) OCCO3
Molecular Formula
C24H25ClN4O3
Molecular Weight
452.93
Storage Conditions
-20°C
Notes
For research use only.
Available Sizes
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