SSTR5 antagonist 3
Compound 23 is a potent, orally active SSTR5 antagonist with low hERG affinity, exhibiting IC50 values of 2.8 nM (human) and 1.4 nM (mouse) . It is a valuable research tool for investigating SSTR5 function in gallstone disease and metabolic disorders, supporting both in vitro binding assays and in vivo pharmacological studies.
Product Specifications
CAS Number
2851454-42-5
Field of Research
Cancer Biology; Pharmacology & Drug Discovery, Pharmacology & Drug Discovery
Smiles
O (CC) C1=C (C (OCC) =CC (CN2CCC (CNC3=CC (OC) =C (C (O) =O) C=C3) (F) CC2) =C1) C4=CC=C (F) C=C4
Molecular Formula
C31H36F2N2O5
Molecular Weight
554.62
Storage Conditions
-20°C
Notes
For research use only.
Available Sizes
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