5-HT6R antagonist 1
Compound 8 (5-HT6R antagonist 1) is a potent serotonin 6 receptor antagonist (K i = 5 nM) with antiplatelet activity and high metabolic stability. It has demonstrated efficacy in reversing cognitive deficits in rodent models of memory impairment, supporting its investigation for Alzheimer's disease-related research.
Product Specifications
Field of Research
Neuroscience, Pharmacology & Drug Discovery
Molecular Formula
C17H22F2N6O
Molecular Weight
364.39
Storage Conditions
-20°C
Notes
For research use only.
Available Sizes
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