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5-HT6R antagonist 1

Compound 8 (5-HT6R antagonist 1) is a potent serotonin 6 receptor antagonist (K i = 5 nM) with antiplatelet activity and high metabolic stability. It has demonstrated efficacy in reversing cognitive deficits in rodent models of memory impairment, supporting its investigation for Alzheimer's disease-related research.

Product Specifications

Field of Research

Neuroscience, Pharmacology & Drug Discovery

Molecular Formula

C17H22F2N6O

Molecular Weight

364.39

Storage Conditions

-20°C

Notes

For research use only.

Available Sizes

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