MS2177
MS2177 is a potent and selective SETD8 inhibitor with a reported IC50 of 1.9 μM and a KD of 1.3 μM. This compound is a valuable chemical probe for studying H4K20 monomethylation in epigenetic research, applicable in both cell-based and biochemical assays to investigate gene regulation and cellular processes.
Product Specifications
Smiles
COC1=C (OCCN) C=C (N=C (N2CCCC2) N=C3NCCCCCN4CCCC4) C3=C1
Molecular Formula
C24H38N6O2
Molecular Weight
442.61
Storage Conditions
-20°C
Notes
For research use only.
Available Sizes
Frequently Asked Questions
More Discoveries
Explore Other Products
Browse additional items from our catalog