Ep300/CREBBP-IN-2
Ep300/CREBBP-IN-2 (Example 73) is a potent, orally bioavailable dual inhibitor of Ep300 and CREBBP with IC50 values of 0.052 μM and 0.148 μM, respectively. It is widely used in cancer research to investigate the roles of these acetyltransferases in tumorigenesis, both in cellular and animal models.
Product Specifications
CAS Number
2259641-59-1
Field of Research
Epigenetics & Chromatin, Signal Transduction
Smiles
COc1ccc (cc1) C1 (CCC (F) (F) CC1) C (=O) N1C[C@H] (F) C[C@@H]1C (=O) Nc1ccc2NC (=O) Cc2n1
Molecular Formula
C26H27F3N4O4
Molecular Weight
516.51
Storage Conditions
-20°C
Notes
For research use only.
Available Sizes
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