Ep300/CREBBP-IN-3
Ep300/CREBBP-IN-3 (Example 61) is a dual inhibitor of the histone acetyltransferases EP300 and CREBBP with IC50 values of 56 nM and 95 nM, respectively. This cell-permeable compound is a valuable chemical probe for epigenetic and cancer research, enabling mechanistic studies in both cellular and biochemical assays.
Product Specifications
CAS Number
2259641-47-7
Field of Research
Epigenetics & Chromatin, Signal Transduction
Smiles
F[C@@H]1C[C@@H] (N (C1) C (=O) C1 (CCCCC1) c1ccc (cc1) C (=O) C (F) (F) F) C (=O) Nc1ccc2[nH]ncc2n1
Molecular Formula
C26H25F4N5O3
Molecular Weight
531.50
Storage Conditions
-20°C
Notes
For research use only.
Available Sizes
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