Ep300/CREBBP-IN-4
Ep300/CREBBP-IN-4 (Example 56) is a potent dual inhibitor of EP300 and CREBBP with IC50 values of 24 nM and 64 nM, respectively. It is a valuable chemical probe for oncology research, used to investigate the roles of these acetyltransferases in cancer cell proliferation and tumorigenesis in both cellular and animal models.
Product Specifications
CAS Number
2259641-42-2
Field of Research
Epigenetics & Chromatin, Signal Transduction
Smiles
COc1ccc (cc1) C1 (CC (F) (F) C1) C (=O) N1C[C@H] (F) C[C@@H]1C (=O) Nc1ccc2[nH]ncc2n1
Molecular Formula
C23H22F3N5O3
Molecular Weight
473.45
Storage Conditions
-20°C
Notes
For research use only.
Available Sizes
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