PROTAC BRD4 Degrader-11
PROTAC BRD4 Degrader-11 is a potent heterobifunctional degrader that effectively targets BRD4 via VHL recruitment, demonstrating high activity in PC3 prostate cancer cells with sub-nanomolar DC50 values. Its utility extends to targeted protein degradation research in oncology, particularly for studying BRD4's role in cancer cell proliferation in vitro.
Product Specifications
Field of Research
Epigenetics & Chromatin, Pharmacology & Drug Discovery
Molecular Formula
C61H75F2N9O12S4
Molecular Weight
1292.56
Storage Conditions
-20°C
Notes
For research use only.
Available Sizes
Frequently Asked Questions
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