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(R) -V-0219 hydrochloride

(R) -V-0219 hydrochloride is the orally bioavailable (R) -enantiomer of V-0219, acting as a positive allosteric modulator (PAM) of the human GLP-1 receptor. It demonstrates functional activity by mobilizing intracellular calcium in hGLP-1R-expressing HEK293 cells, supporting its use in metabolic disease research.

Product Specifications

Field of Research

Pharmacology & Drug Discovery

Molecular Formula

C20H26ClF3N4O2

Molecular Weight

446.89

Storage Conditions

-20°C

Notes

For research use only.

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