PDK-IN-1
PDK-IN-1 (compound 7o) is a dual inhibitor of pyruvate dehydrogenase kinase (PDK1) and HSP90 with IC50 values of 0.03 μM and 0.1 μM, respectively. It targets the PDH/PDK axis and has demonstrated significant antitumor efficacy by reducing tumor mass in in vivo studies.
Product Specifications
CAS Number
2897696-10-3
Field of Research
Metabolism Research, Signal Transduction
Smiles
CN1C=C (C=2C1=NC=C (Br) C2) C=3C (=NN=C (N) N3) C=4C=5C (NC4) =CC=C (OC) C5
Molecular Formula
C20H16BrN7O
Molecular Weight
450.29
Storage Conditions
-20°C
Notes
For research use only.
Available Sizes
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