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LSD1-IN-26

LSD1-IN-26 (12u) is a potent and selective LSD1 inhibitor (IC50 = 25.3 nM) with weaker activity against MAO-A/B. It potently induces apoptosis in MGC-803 gastric cancer cells in vitro, making it a useful chemical probe for oncology research, particularly in studying gastric cancer mechanisms.

Product Specifications

Field of Research

Cell Biology, Epigenetics & Chromatin, Metabolism Research, Neuroscience, Protein Biochemistry

Molecular Formula

C27H25Cl2F2N3O

Molecular Weight

516.41

Storage Conditions

-20°C

Notes

For research use only.

Available Sizes

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