Nampt degrader-2
Nampt degrader-2 is a fluorescent PROTAC molecule that induces degradation of NAMPT via the VHL E3 ligase, with an IC50 of 41.9 nM. This degradation depletes cellular NAD+ and demonstrates potent antitumor activity in research models, supporting its use in oncology and metabolic studies.
Product Specifications
Field of Research
Metabolism Research, Pharmacology & Drug Discovery
Molecular Formula
C59H73N9O7S
Molecular Weight
1052.33
Storage Conditions
-20°C
Notes
For research use only.
Available Sizes
Frequently Asked Questions
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